SCHEMBL177582

SCHEMBL177582

OB(O)c1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
HTR3A P46098 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
KDR P35968 1/20 0.47
MGLL Q99685 2/20 0.47
TTR P02766 1/20 0.46
IDO1 P14902 2/20 0.43
PDK1 Q15118 1/20 0.42
NPFFR2 Q9Y5X5 3/20 0.41
NPFFR1 Q9GZQ6 2/20 0.41
ENPP2 Q13822 1/20 0.41
NOTUM Q6P988 5/20 0.41
LMNA P02545 1/20 0.40
RAPGEF4 Q8WZA2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29465748 1.00 HTR3E (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL17196033 0.85 TTR (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL177526 0.84 TTR (0.50) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL257875 0.81 CA1 (0.47) KDRMGLLIDO1
SCHEMBL3789433 0.81 MGLL (0.52) MGLLTTRENPP2
SCHEMBL29700447 0.81 MGLL (0.52) MGLLTTRENPP2
SCHEMBL29525231 0.78 MGLL (0.48) MGLLENPP2
SCHEMBL7895094 0.78 MGLL (0.48) MGLLTTRENPP2LMNA
SCHEMBL206793 0.78 MGLL (0.48) MGLLENPP2
SCHEMBL23229016 0.77 IDO1 (0.42) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 369 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116874534-A Carboxamide group-based ionic iridium (III) complex, preparation method thereof and application thereof in fluoride ion detection 桂林理工大学 2023-10-13 CN claimed
EP-3478673-B1 CYANOINDOLINE DERIVATIVES AS NIK INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2020-09-16 EP claimed
EP-2948453-B1 PYRAZOLO[3,4-D]PYRIMIDINONE COMPOUNDS AS INHIBITORS OF THE P53/MDM2 INTERACTION NOVARTIS AG (CH) 2017-08-02 EP claimed
EP-2948451-B1 SUBSTITUTED PURINONE COMPOUNDS NOVARTIS AG (CH) 2017-07-12 EP claimed
EP-2018371-B1 PRIMARY AMINES AND DERIVATIVES THEREOF AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARM INC (US) 2015-03-04 EP claimed
EP-1928875-B1 2-amino-7,8-dihydro-6H-pyrido(4,3-d)pyrimidin-5-ones, process for their preparation and pharmaceutical compositions containing the same NOVARTIS AG (CH) 2011-06-29 EP claimed
EP-4719385-A2 1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINES AS ANTI-INFECTIOUS AGENTS University of Vermont and State Agricultural College (US) 2026-04-08 EP disclosed
US-20260035360-A1 INHIBITORS OF MYC AND USES THEREOF UNIV NORTHWESTERN (US) 2026-02-05 US disclosed
US-20250257064-A1 TRIFLUOROMETHYL-SUBSTITUTED SULFONAMIDE AS BCL-2-SELECTIVE INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2025-08-14 US disclosed
US-12371431-B2 Trifluoromethyl-substituted sulfonamide as BCL-2-selective inhibitor CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2025-07-29 US disclosed
EP-4561568-A2 INHIBITORS OF MYC AND USES THEREOF Northwestern University (US) 2025-06-04 EP disclosed
CN-116472266-B Compounds as prolyl hydroxylase inhibitors and methods of making the same 苏中药业集团股份有限公司 2025-05-30 CN disclosed
WO-2025076088-A1 LACTAMS FOR USE AS SARM1 INHIBITORS GENENTECH, INC. (US) 2025-04-10 WO disclosed
US-5578724-A INHIBITORS OF 5-ALPHA-REDUCTASE ELI LILLY AND COMPANY (US) 1996-11-26 US disclosed
WO-1996035422-A1 METHODS FOR INHIBITING BONE LOSS ELI LILLY AND COMPANY (US) 1996-11-14 WO disclosed
EP-0742010-A2 Benzoquinolin-3-ones to inhibit bone loss ELI LILLY AND COMPANY (US) 1996-11-13 EP disclosed
EP-0733365-A2 Use of benzoquinolin-3-ones for the treatment and prevention of prostatic cancer ELI LILLY AND COMPANY (US) 1996-09-25 EP disclosed
US-5550134-A ADMINISTERING TO A MAMMAL FROM A SERIES OF BENZOQUINOLIN-3-ONE COMPOUNDS ELI LILLY AND COMPANY (US) 1996-08-27 US disclosed
WO-1996009046-A1 5α-REDUCTASE INHIBITORS ELI LILLY AND COMPANY (US) 1996-03-28 WO disclosed
EP-0703221-A1 5 alpha-reductase Inhibitors ELI LILLY AND COMPANY (US) 1996-03-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12371431-B2 Trifluoromethyl-substituted sulfonamide as BCL-2-selective inhibitor BCL2L11, BCL2, BCL2L2 HTR3E 4313/4885HTR3B 3917/4885HTR3A 4519/4885
US-20260035360-A1 INHIBITORS OF MYC AND USES THEREOF MYC, MYCBP, MYCBP2 HTR3E 2506/4885HTR3B 3311/4885HTR3A 3130/4885
US-20250257064-A1 TRIFLUOROMETHYL-SUBSTITUTED SULFONAMIDE AS BCL-2-SELECTIVE INHIBITOR BCL2, BAX, BCL2L2 HTR3E 3932/4885HTR3B 3635/4885HTR3A 4347/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.