SCHEMBL17761016

SCHEMBL17761016

NC(=O)c1csc(C(=O)N2CCSCC2)n1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.46
RAB9A P51151 1/20 0.46
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HRH3 Q9Y5N1 1/20 0.37
HTR2B P41595 1/20 0.37
HTR2C P28335 2/20 0.36
KMT2A Q03164 1/20 0.36
CYP2C19 P33261 1/20 0.34
ACHE P22303 1/20 0.34
CNR2 P34972 1/20 0.34
TRPC3 Q13507 2/20 0.33
TRPC6 Q9Y210 2/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31240238 0.88 HTR2C (0.42) HPGDRAB9AALDH1A1HSD17B10HRH3
SCHEMBL17711525 0.86 HPGD (0.47) HPGDRAB9AALDH1A1HSD17B10HTR2C
SCHEMBL28176249 0.84 HTR2C (0.52) HPGDRAB9AHRH3HTR2C
SCHEMBL28580100 0.79 MAPT (0.41) HPGDRAB9AALDH1A1HSD17B10HRH3
SCHEMBL17711415 0.78 HPGD (0.40) HPGDRAB9AALDH1A1HSD17B10HTR2C
SCHEMBL2745784 0.74 HTR2B (0.49) RAB9AALDH1A1HRH3HTR2BKMT2A
SCHEMBL12169124 0.71 HTR2B (0.50) ALDH1A1HTR2BCYP2C19ACHE
SCHEMBL17076771 0.71 HTR2B (0.35) HRH3HTR2BCYP2C19ACHE
SCHEMBL15012294 0.70 HTR2C (0.53) HPGDRAB9AHRH3HTR2C
SCHEMBL12188683 0.70 SCD5 (0.44) HRH3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3212643-A1 TRIFLUOROMETHYL ALCOHOLS AS MODULATORS OF RORyt Janssen Pharmaceutica, N.V. (BE) 2017-09-06 EP disclosed
WO-2016069974-A1 TRIFLUOROMETHYL ALCOHOLS AS MODULATORS OF RORyt JANSSEN PHARMACEUTICA NV (BE) 2016-05-06 WO disclosed