SCHEMBL1776252

SCHEMBL1776252

Cc1onc(-c2ccccn2)c1COc1ccc(C(=O)NC(C)(C)CO)nn1

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 9/20 0.70
ITGA5 P08648 2/20 0.67
GABRA5 P31644 10/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1777284 0.89 GABRA5 (0.75) GABRA1ITGA5GABRA5
SCHEMBL1776180 0.88 GABRA1 (0.79) GABRA1GABRA5
SCHEMBL1777110 0.87 ITGA5 (0.73) GABRA1ITGA5GABRA5
SCHEMBL1776588 0.86 ITGA5 (0.72) GABRA1ITGA5GABRA5
SCHEMBL1778385 0.86 GABRA1 (0.70) GABRA1ITGA5GABRA5
SCHEMBL2922915 0.86 GABRA5 (0.79) ITGA5GABRA5
SCHEMBL288158 0.86 GABRA5 (0.55) GABRA1ITGA5GABRA5
SCHEMBL1777385 0.85 ITGA5 (0.71) GABRA1ITGA5GABRA5
SCHEMBL1776995 0.85 GABRA5 (0.73) GABRA1ITGA5GABRA5
SCHEMBL1777103 0.84 GABRA5 (0.76) GABRA1ITGA5GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943619-B2 Isoxazolo-pyridazine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-17 US claimed
US-7943619-B2 Isoxazolo-pyridazine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-17 US disclosed