SCHEMBL17772011

SCHEMBL17772011

C[C@@H]1[C@@H](c2ccc(Br)cc2)C1(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
POLB P06746 1/20 0.41
HSD17B10 Q99714 1/20 0.39
CYP2A6 P11509 1/20 0.38
KDM1A O60341 6/20 0.37
RCOR1 Q9UKL0 3/20 0.37
KCNH2 Q12809 2/20 0.37
MAOB P27338 2/20 0.37
KDM1B Q8NB78 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GAA P10253 2/20 0.35
CYP3A4 P08684 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP2C19 P33261 2/20 0.33
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
KMT2A Q03164 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4324752 0.79 ALDH1A1 (0.43) TSHRHSD17B10CYP2A6KDM1ARCOR1
SCHEMBL18898525 0.76 RECQL (0.41) POLBKDM1ARCOR1GAAHSD11B1
SCHEMBL10975565 0.75 CHRNA7 (0.47) KDM1AMAOBALDH1A1CYP2C19MEN1
SCHEMBL17346807 0.73 GAA (0.37) TSHRPOLBHSD17B10CYP2A6KDM1A
SCHEMBL16819947 0.73 HSD17B10 (0.38) TSHRPOLBHSD17B10CYP2A6KDM1A
SCHEMBL15559251 0.73 GAA (0.37) TSHRPOLBHSD17B10CYP2A6KDM1A
SCHEMBL16841716 0.73 HSD17B10 (0.38) TSHRPOLBHSD17B10CYP2A6KDM1A
SCHEMBL16819998 0.73 GAA (0.37) TSHRPOLBHSD17B10CYP2A6KDM1A
SCHEMBL15442881 0.71 SLC9A1 (0.45) TSHRHSD17B10LMNAKMT2A
SCHEMBL15442883 0.71 SLC9A1 (0.45) TSHRHSD17B10LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2670731-B1 POSITIVE ALLOSTERIC MODULATORS OF THE ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR AND USES THEREOF. BIONOMICS LTD (AU) 2016-05-25 EP disclosed