SCHEMBL17782865

SCHEMBL17782865

N#Cc1ccc(C(F)(F)F)cc1S

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AR P10275 11/20 0.49
TRPV4 Q9HBA0 3/20 0.44
KIF11 P52732 2/20 0.44
TAS2R14 Q9NYV8 1/20 0.43
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
PTPN1 P18031 1/20 0.40
PTPN6 P29350 1/20 0.40
PTPN11 Q06124 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29224606 0.98 AR (0.47) ARTRPV4KIF11TAS2R14CYP11B1
SCHEMBL30945835 0.98 AR (0.47) ARTRPV4KIF11TAS2R14CYP11B1
SCHEMBL3480548 0.85 KIF11 (0.56) ARKIF11CYP11B1CYP11B2
SCHEMBL29546917 0.83 AR (0.52) ARKIF11TAS2R14CYP11B1CYP11B2
SCHEMBL12151755 0.83 AR (0.52) ARKIF11TAS2R14CYP11B1CYP11B2
SCHEMBL495426 0.79 CYP11B1 (0.57) ARTRPV4KIF11TAS2R14CYP11B1
SCHEMBL1996075 0.79 AR (0.73) AR
SCHEMBL964361 0.79 AR (0.49) ARKIF11TAS2R14
SCHEMBL16952881 0.78 AR (0.47) ARKIF11TAS2R14CYP11B1CYP11B2
SCHEMBL669827 0.78 AR (0.47) ARKIF11TAS2R14CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118146127-A Preparation method of 2-methylthio-4-trifluoromethyl benzonitrile 北京颖泰嘉和生物科技股份有限公司 2024-06-07 CN disclosed
WO-2022015624-A1 SUBSTITUTED DIHYDROPYRAZINEDIONES AS MODULATORS OF THE NMDA RECEPTOR SCHRÖDINGER, INC. (US) 2022-01-20 WO disclosed
CN-109111405-B Aromatic thioether compound and pesticide and medical application thereof 南开大学 2021-07-30 CN disclosed
US-9662328-B2 Targeting human thymidylate kinase induces DNA repair toxicity in malignant tumor cells NATIONAL TAIWAN UNIVERSITY (TW) 2017-05-30 US disclosed
CN-106565621-A Isoxaflutole synthesizing method 上虞颖泰精细化工有限公司 2017-04-19 CN disclosed
US-20160151362-A1 TARGETING HUMAN THYMIDYLATE KINASE INDUCES DNA REPAIR TOXICITY IN MALIGNANT TUMOR CELLS NATIONAL TAIWAN UNIVERSITY (TW) 2016-06-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160151362-A1 TARGETING HUMAN THYMIDYLATE KINASE INDUCES DNA REPAIR TOXICITY IN MALIGNANT TUMOR CELLS DTYMK, TYMP, TK1 AR 4387/4885TRPV4 4115/4885KIF11 2850/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.