SCHEMBL17786233

SCHEMBL17786233

CCOC(=O)N1CCN(Cc2nc3c(c(=O)n(C)c(=O)n3C)n2CCC(C)C)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 17/20 1.00
KMT2A Q03164 2/20 1.00
HSD17B10 Q99714 3/20 0.81
TP53 P04637 1/20 0.81
LMNA P02545 2/20 0.79
TSHR P16473 4/20 0.70
SMN1; SMN2 Q16637 2/20 0.70
ALOX15 P16050 2/20 0.70
USP2 O75604 4/20 0.69
CASP1 P29466 1/20 0.68
CASP7 P55210 1/20 0.68
MEN1 O00255 1/20 0.67
L3MBTL1 Q9Y468 1/20 0.66
NPSR1 Q6W5P4 2/20 0.65
HTT P42858 1/20 0.65
GAA P10253 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17791583 0.87 ALDH1A1 (0.81) ALDH1A1KMT2AHSD17B10TP53LMNA
SCHEMBL17786260 0.85 ALDH1A1 (0.75) ALDH1A1KMT2AHSD17B10TP53LMNA
SCHEMBL17791573 0.85 ALDH1A1 (0.75) ALDH1A1KMT2AHSD17B10TP53LMNA
SCHEMBL17786253 0.84 ALDH1A1 (1.00) ALDH1A1KMT2AHSD17B10TP53LMNA
SCHEMBL17791580 0.81 ALDH1A1 (0.72) ALDH1A1KMT2AHSD17B10TP53LMNA
SCHEMBL17791591 0.81 HSD17B10 (1.00) ALDH1A1KMT2AHSD17B10TP53LMNA
SCHEMBL17786264 0.81 ALDH1A1 (0.93) ALDH1A1KMT2AHSD17B10TP53LMNA
SCHEMBL17791575 0.81 ALDH1A1 (0.70) ALDH1A1KMT2AHSD17B10TP53LMNA
SCHEMBL17207521 0.80 ALDH1A1 (1.00) ALDH1A1KMT2AHSD17B10TP53TSHR
SCHEMBL17791863 0.80 ALDH1A1 (0.84) ALDH1A1KMT2AHSD17B10TP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016086008-A1 SMALL MOLECULE ALDEHYDE DEHYDROGENASE INHIBITORS AND METHODS OF USE THEREOF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2016-06-02 WO disclosed
WO-2016086008-A1 SMALL MOLECULE ALDEHYDE DEHYDROGENASE INHIBITORS AND METHODS OF USE THEREOF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2016-06-02 WO disclosed