SCHEMBL1778735

SCHEMBL1778735

CCC(=O)N1CCSCC1n1c(-c2cc3cccnc3[nH]2)cc2cc(OC)ccc21

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 14/20 0.41
CCNB2 O95067 1/20 0.41
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39
IGF1R P08069 1/20 0.34
CALCRL Q16602 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1778731 0.83 RIPK1 (0.39) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1779933 0.77 DRD2 (0.44) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1777680 0.73 RIPK1 (0.60) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1778988 0.72 RIPK1 (0.49) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1777852 0.71 RIPK1 (0.49) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1778783 0.70 RIPK1 (0.48) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1778695 0.69 RIPK1 (0.46) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1779504 0.69 IGF1R (0.47) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1777443 0.69 RIPK1 (0.46) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL1778453 0.68 RIPK1 (0.45) RIPK1CCNB2CDK1CCNB1CCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943616-B2 Protein kinase inhibitors; astham; psoriasis; antiinflammatory agents; inflammatory bowel disorders AVENTIS PHARMACEUTICALS INC. (US) 2011-05-17 US disclosed
EP-1397360-A1 AZAINDOLES Aventis Pharma Limited (GB) 2004-03-17 EP disclosed
WO-2003000688-A1 AZAINDOLES AVENTIS PHARMA LIMITED (GB) 2003-01-03 WO disclosed