SCHEMBL17801727

SCHEMBL17801727

CCCCOC(=O)N1CCCc2cc(NC(=O)OCc3ccccc3)ccc2C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 16/20 0.56
SIGMAR1 Q99720 16/20 0.56
ALDH1A1 P00352 1/20 0.46
TMPRSS2 O15393 1/20 0.45
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
DRD1 P21728 1/20 0.44
HRH2 P25021 1/20 0.44
HTR1B P28222 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR1E P28566 1/20 0.44
SLC6A4 P31645 1/20 0.44
HRH1 P35367 1/20 0.44
HTR2B P41595 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17797697 0.85 TMEM97 (0.55) TMEM97SIGMAR1ALDH1A1TMPRSS2NPC1
SCHEMBL6292442 0.84 TMEM97 (0.62) TMEM97SIGMAR1ALDH1A1TMPRSS2HTR1A
SCHEMBL17797565 0.81 TMEM97 (0.54) TMEM97SIGMAR1ALDH1A1NPC1TP53
SCHEMBL17797552 0.81 TMEM97 (0.55) TMEM97SIGMAR1ALDH1A1NPC1TP53
SCHEMBL6296029 0.80 TMEM97 (0.62) TMEM97SIGMAR1ALDH1A1TMPRSS2HTR1A
SCHEMBL2181843 0.79 ESR2 (0.58) TMEM97SIGMAR1ALDH1A1TMPRSS2NPC1
SCHEMBL6296040 0.79 TMPRSS2 (0.56) TMEM97SIGMAR1ALDH1A1TMPRSS2NPC1
SCHEMBL17797663 0.78 TMEM97 (0.55) TMEM97SIGMAR1ALDH1A1HTR1AADRA2A
SCHEMBL9447608 0.78 NPC1 (0.65) ALDH1A1NPC1TP53MAPTNFKB1
SCHEMBL17813396 0.77 PSEN1 (0.49) TMEM97SIGMAR1ALDH1A1HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016090079-A1 HETEROARYL COMPOUNDS AND USES THEREOF CELGENE AVILOMICS RESEARCH, INC. (US) 2016-06-09 WO disclosed