SCHEMBL17801744

SCHEMBL17801744

O=C(O)Oc1ccc2nc(-c3cncc(F)c3)sc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 6/20 0.49
PIK3CG P48736 1/20 0.47
DYRK1A Q13627 4/20 0.44
SULT1A1 P50225 2/20 0.43
KDM4E B2RXH2 2/20 0.43
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CLK1 P49759 1/20 0.43
CLK2 P49760 1/20 0.43
DYRK2 Q92630 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
KMT2A Q03164 1/20 0.41
CA2 P00918 1/20 0.41
NPC1 O15118 1/20 0.41
MITF O75030 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16568908 0.83 KDM4E (0.64) APPPIK3CGDYRK1ASULT1A1KDM4E
SCHEMBL17801689 0.82 NPC1 (0.56) PIK3CGKDM4ENFKB1NFKB2RELA
SCHEMBL17801701 0.76 APP (0.69) APPSULT1A1KDM4ENFKB1NFKB2
Hydrochloric Acid SCHEMBL22130203 0.75 APP (0.68) APPSULT1A1KDM4ENFKB1NFKB2
SCHEMBL20068806 0.73 DYRK1A (0.63) APPDYRK1AKDM4ENFKB1NFKB2
SCHEMBL16568922 0.71 HDAC6 (0.46) PIK3CGDYRK1AKDM4ENFKB1NFKB2
SCHEMBL11024521 0.71 KMT2A (0.57) DYRK1ASMN1; SMN2KMT2ACA2NPC1
SCHEMBL9620877 0.70 CA2 (0.56) APPSULT1A1KDM4ESMN1; SMN2KMT2A
SCHEMBL5760456 0.70 MAPT (0.48) APPDYRK1AKDM4EKMT2ACA2
SCHEMBL3042970 0.69 APP (0.70) APPSULT1A1KDM4ENFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3227283-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS Bayer CropScience AG (DE) 2017-10-11 EP disclosed
WO-2016087371-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-06-09 WO disclosed