SCHEMBL17801978

SCHEMBL17801978

O=[N+]([O-])c1cccc2c1OCCN(CC1CC1)C2

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 4/20 0.40
GRM2 Q14416 1/20 0.39
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
SIGMAR1 Q99720 1/20 0.38
ACHE P22303 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17802004 0.84 KMT2A (0.41) ACKR3CHRNB4CHRNA3CYP1A2CYP2D6
SCHEMBL17801946 0.81 ACKR3 (0.42) ACKR3GRM2CHRNB4CHRNA3SIGMAR1
SCHEMBL19582241 0.81 ACKR3 (0.43) ACKR3CYP1A2CYP2D6CYP2C19
SCHEMBL17801898 0.77 GRM2 (0.43) ACKR3GRM2CHRNB4CHRNA3ACHE
SCHEMBL19582257 0.76 ACKR3 (0.40) ACKR3GRM2SIGMAR1ACHECYP1A2
SCHEMBL19582463 0.75 GRM2 (0.50) ACKR3GRM2CHRNB4CHRNA3ACHE
SCHEMBL17801896 0.72 ACKR3 (0.57) ACKR3
SCHEMBL8948801 0.71 PARP1 (0.49) ACHEKMT2A
SCHEMBL10659420 0.68 ALDH1A1 (0.42) CHRNB4CHRNA3ACHEMEN1KMT2A
SCHEMBL17802010 0.68 GRM2 (0.50) ACKR3GRM2CHRNB4CHRNA3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3227263-A1 CXCR7 RECEPTOR MODULATORS Actelion Pharmaceuticals Ltd (CH) 2017-10-11 EP disclosed
WO-2016087370-A1 CXCR7 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-06-09 WO disclosed