SCHEMBL17804167

SCHEMBL17804167

C=C(O)c1ccnc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.45
TRPA1 O75762 1/20 0.41
LOX P28300 1/20 0.41
LOXL3 P58215 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
TAS1R3 Q7RTX0 2/20 0.39
TAS1R1 Q7RTX1 2/20 0.39
TAS1R2 Q8TE23 2/20 0.39
IDO1 P14902 1/20 0.38
SMARCA2 P51531 2/20 0.37
SMARCA4 P51532 2/20 0.37
KDM4E B2RXH2 1/20 0.36
KDM6B O15054 1/20 0.36
TET3 O43151 1/20 0.36
KDM4A O75164 1/20 0.36
BBOX1 O75936 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
KDM5A P29375 1/20 0.36
KDM5C P41229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30820861 0.81 RECQL (0.44) RECQLTRPA1LOXLOXL3LOXL2
SCHEMBL5700002 0.81 RECQL (0.44) RECQLTRPA1LOXLOXL3LOXL2
SCHEMBL13742411 0.81 RECQL (0.44) RECQLTRPA1LOXLOXL3LOXL2
SCHEMBL40123 0.78 KDM4C (0.61) RECQLTAS1R3TAS1R1TAS1R2KDM4E
Bromide SCHEMBL7842108 0.77 KDM4C (0.59) RECQLTAS1R3TAS1R1TAS1R2KDM4E
Hydrochloric Acid SCHEMBL7221156 0.77 KDM4C (0.59) RECQLTAS1R3TAS1R1TAS1R2KDM4E
SCHEMBL31547893 0.77 KDM4C (0.59) RECQLTAS1R3TAS1R1TAS1R2KDM4E
Methane SCHEMBL9122275 0.77 KDM5C (0.59) RECQLTAS1R3TAS1R1TAS1R2KDM4E
SCHEMBL15391333 0.76 RECQL (0.40) RECQLTRPA1LOXLOXL3LOXL2
SCHEMBL27623752 0.76 RECQL (0.47) RECQLLOXLOXL3LOXL2TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3029031-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2016-06-08 EP disclosed