SCHEMBL17804350

SCHEMBL17804350

CCCC(=O)c1cc(Br)cc(N(C)C2CCOCC2)c1C

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EZH2 Q15910 14/20 0.55
EED O75530 1/20 0.44
RBBP4 Q09028 1/20 0.44
SUZ12 Q15022 1/20 0.44
AEBP2 Q6ZN18 1/20 0.44
EZH1 Q92800 1/20 0.44
PDE4B Q07343 3/20 0.36
PDE4D Q08499 3/20 0.35
PDE4A P27815 2/20 0.35
PDE4C Q08493 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18829901 0.84 EZH2 (0.57) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL13280225 0.84 EZH2 (0.57) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL13276998 0.81 EZH2 (0.56) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL17804325 0.76 EZH2 (0.42) EZH2PDE4ANPC1MEN1KMT2A
SCHEMBL17804355 0.76 EZH2 (0.41) EZH2
SCHEMBL13277238 0.74 EZH2 (0.51) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL18829912 0.74 EZH2 (0.60) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL13276540 0.74 EZH2 (0.60) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL29613562 0.74 EZH2 (0.60) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL30499098 0.73 EZH2 (0.59) EZH2EEDRBBP4SUZ12AEBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697198-B1 SUBSTITUTED BENZENE COMPOUNDS EPIZYME INC (US) 2016-06-08 EP disclosed