SCHEMBL178077

SCHEMBL178077

BrC(I)CCCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
ALOX12 P18054 1/20 0.46
CASP1 P29466 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SIGMAR1 Q99720 3/20 0.45
MAOA P21397 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
MAOB P27338 2/20 0.43
HTR2A P28223 1/20 0.43
KCNH2 Q12809 1/20 0.43
GRIK1 P39086 1/20 0.42
IDO1 P14902 1/20 0.42
HDAC3 O15379 1/20 0.42
MAPK1 P28482 1/20 0.42
ADRA1A P35348 1/20 0.42
HDAC4 P56524 1/20 0.42
SLC6A3 Q01959 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6682085 0.82 SIGMAR1 (0.48) SIGMAR1MAOATDP1MAOBHTR2A
SCHEMBL8325572 0.78 SIGMAR1 (0.47) ALDH1A1HPGDALOX15ALOX12CASP1
SCHEMBL29029777 0.78 MAOA (0.50) ALDH1A1HPGDALOX15ALOX12CASP1
SCHEMBL1487691 0.78 MAOB (0.48) SIGMAR1MAOB
SCHEMBL10991606 0.78 SIGMAR1 (0.45) SIGMAR1MAOATDP1MAOBHTR2A
SCHEMBL9347969 0.77 MAOB (0.45) SIGMAR1MAOATDP1MAOBHTR2A
SCHEMBL6686320 0.76 MAOA (0.52) SIGMAR1MAOATDP1MAOB
SCHEMBL1128437 0.75 SIGMAR1 (0.46) SIGMAR1MAOATDP1KCNH2ADRA1A
Bromide SCHEMBL10928757 0.75 SIGMAR1 (0.50) SIGMAR1MAOAMAOBHTR2AKCNH2
SCHEMBL1678945 0.74 GRIK1 (0.54) ALDH1A1HPGDGRIK1HDAC3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399585-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2011-12-28 EP disclosed