SCHEMBL17814060

SCHEMBL17814060

CC(=O)N(c1ccccc1)C1CCN(Cc2nc(-c3ccc(Cl)c(Cl)c3)[nH]c2C)CC1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.58
CHRM2 P08172 3/20 0.48
CHRM3 P20309 3/20 0.48
OPRM1 P35372 1/20 0.44
SIGMAR1 Q99720 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20861032 0.90 CTSS (0.57) CTSSOPRM1
SCHEMBL6654442 0.81 CTSS (0.49) CTSSCHRM2CHRM3OPRM1SIGMAR1
SCHEMBL20861268 0.81 CTSS (0.57) CTSS
SCHEMBL17813969 0.81 CTSS (0.58) CTSS
SCHEMBL6652795 0.80 DRD2 (0.51) CTSSCHRM2CHRM3OPRM1SIGMAR1
SCHEMBL6653716 0.79 DRD2 (0.50) CTSSCHRM2CHRM3OPRM1SIGMAR1
SCHEMBL6649677 0.79 CTSS (0.47) CTSSOPRM1SIGMAR1
SCHEMBL6653777 0.76 CTSS (0.57) CTSS
SCHEMBL20861218 0.75 CTSS (0.59) CTSS
SCHEMBL20861229 0.74 CTSS (0.49) CTSSOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016087352-A1 NOVEL PIPERIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2016-06-09 WO disclosed