SCHEMBL17814697

SCHEMBL17814697

CCOc1ccc(Nc2nc(=O)c3c(ncn3CC)n2Cc2ccc(Cl)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 19/20 0.57
BRD4 O60885 1/20 0.51
BRD2 P25440 1/20 0.51
BRD3 Q15059 1/20 0.51
BRDT Q58F21 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814723 0.91 BRD4 (0.48) P2RX3BRD4BRD2BRD3BRDT
SCHEMBL17814696 0.90 P2RX3 (0.55) P2RX3BRD4BRD2BRD3BRDT
SCHEMBL17814730 0.90 P2RX3 (0.64) P2RX3
SCHEMBL17814695 0.90 P2RX3 (0.56) P2RX3BRD4BRD2BRD3BRDT
SCHEMBL17814743 0.89 P2RX3 (0.57) P2RX3
SCHEMBL17814694 0.89 P2RX3 (0.55) P2RX3BRD4BRD2BRD3BRDT
SCHEMBL17814686 0.88 BRD4 (0.53) P2RX3BRD4BRD2BRD3BRDT
SCHEMBL19682490 0.88 P2RX3 (0.55) P2RX3
SCHEMBL19682703 0.88 P2RX3 (0.66) P2RX3
SCHEMBL17814744 0.87 P2RX3 (0.51) P2RX3BRD4BRD2BRD3BRDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017209267-A1 PURINE DERIVATIVE 塩野義製薬株式会社 2017-12-07 WO disclosed
WO-2016088838-A1 PURINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION THEREOF 塩野義製薬株式会社 2016-06-09 WO disclosed