SCHEMBL17814709

SCHEMBL17814709

CSc1nc(=O)c2[nH]cnc2n1Cc1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.54
ATM Q13315 1/20 0.51
APOBEC3G Q9HC16 1/20 0.51
PDE4A P27815 2/20 0.45
PDE4B Q07343 2/20 0.45
PDE4C Q08493 2/20 0.45
PDE4D Q08499 2/20 0.45
MPO P05164 1/20 0.44
TPO P07202 1/20 0.44
ACP1 P24666 1/20 0.43
KMT2A Q03164 2/20 0.42
P2RX7 Q99572 2/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA2B P29275 1/20 0.42
P2RX3 P56373 1/20 0.41
NPC1 O15118 1/20 0.41
TLR7 Q9NYK1 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814735 0.81 PNP (0.57) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL562099 0.75 ADORA2B (0.59) PDE4APDE4BPDE4CPDE4DADORA3
SCHEMBL28911354 0.74 PNP (0.35) PNPATMAPOBEC3GPDE4APDE4B
SCHEMBL17814682 0.74 BRD4 (0.60) ATMAPOBEC3GKMT2AP2RX3MEN1
SCHEMBL7681629 0.73 PNP (0.80) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL3241382 0.72 PDE4A (0.71) PDE4APDE4BPDE4CPDE4DADORA3
SCHEMBL30804835 0.71 ATM (0.52) ATMAPOBEC3GKMT2AP2RX3MEN1
SCHEMBL17814707 0.71 ATM (0.49) ATMAPOBEC3GKMT2AMEN1ALDH1A1
SCHEMBL9983147 0.71 ATM (0.60) ATMAPOBEC3GKMT2AP2RX3TLR7
SCHEMBL7682667 0.71 PNP (0.60) PNPPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409331-B Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-20 CN disclosed
CN-112409331-A Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-02-26 CN disclosed
WO-2017209267-A1 PURINE DERIVATIVE 塩野義製薬株式会社 2017-12-07 WO disclosed
WO-2016088838-A1 PURINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION THEREOF 塩野義製薬株式会社 2016-06-09 WO disclosed