SCHEMBL17814735

SCHEMBL17814735

O=c1nc(S)n(Cc2ccc(Cl)cc2)c2nc[nH]c12

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.57
MPO P05164 1/20 0.46
TPO P07202 1/20 0.46
ACP1 P24666 1/20 0.46
P2RX7 Q99572 2/20 0.42
ADORA3 P0DMS8 1/20 0.41
ADORA2B P29275 1/20 0.41
PDE4A P27815 2/20 0.41
PDE4B Q07343 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
NPC1 O15118 1/20 0.41
KMT2A Q03164 1/20 0.41
TRPA1 O75762 1/20 0.40
TLR7 Q9NYK1 2/20 0.39
TLR8 Q9NR97 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814709 0.81 PNP (0.54) PNPMPOTPOACP1P2RX7
SCHEMBL7681629 0.76 PNP (0.80) PNPMPOTPOACP1ADORA3
SCHEMBL7682667 0.74 PNP (0.60) PNPMPOTPOACP1ADORA3
SCHEMBL17814738 0.73 TNF (0.42) KMT2ATLR7TLR8
SCHEMBL28543435 0.73 PNP (0.37) PNPACP1ADORA3NPC1
SCHEMBL3241382 0.72 PDE4A (0.71) ADORA3ADORA2BPDE4APDE4BPDE4C
SCHEMBL3308563 0.71 PNP (0.51) PNPMPOTPOACP1ADORA3
SCHEMBL17814737 0.69 ALDH1A1 (0.41) KMT2ATLR7TLR8
SCHEMBL30804819 0.68 BRD4 (0.42) KMT2ATLR7TLR8
SCHEMBL29084974 0.68 MPO (0.61) PNPMPOTPOADORA3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409331-B Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-20 CN disclosed
CN-112409331-A Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-02-26 CN disclosed
WO-2017209267-A1 PURINE DERIVATIVE 塩野義製薬株式会社 2017-12-07 WO disclosed
WO-2016088838-A1 PURINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION THEREOF 塩野義製薬株式会社 2016-06-09 WO disclosed