SCHEMBL17822173

SCHEMBL17822173

CCCC(C)NC(=O)C=Cc1ccc(OC)c(OC)c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.73
TAS1R3 Q7RTX0 2/20 0.73
TAS1R1 Q7RTX1 2/20 0.73
NFE2L2 Q16236 1/20 0.60
HPGD P15428 4/20 0.57
LMNA P02545 1/20 0.57
HTT P42858 1/20 0.57
RECQL P46063 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
NPC1 O15118 1/20 0.55
STAT1 P42224 1/20 0.55
RAB9A P51151 1/20 0.55
APP P05067 1/20 0.55
KDM4E B2RXH2 2/20 0.55
ALOX15 P16050 1/20 0.55
MAPK1 P28482 1/20 0.55
HSD17B10 Q99714 1/20 0.55
MMP2 P08253 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17822171 1.00 ALDH1A1 (0.73) ALDH1A1TAS1R3TAS1R1NFE2L2HPGD
SCHEMBL702350 0.89 TAS1R3 (0.70) ALDH1A1TAS1R3TAS1R1NFE2L2HPGD
SCHEMBL702349 0.89 TAS1R3 (0.70) ALDH1A1TAS1R3TAS1R1NFE2L2HPGD
SCHEMBL13002011 0.85 ALDH1A1 (0.70) ALDH1A1TAS1R3TAS1R1NFE2L2HPGD
SCHEMBL703146 0.85 ALDH1A1 (1.00) ALDH1A1TAS1R3TAS1R1HPGDLMNA
SCHEMBL703147 0.85 ALDH1A1 (1.00) ALDH1A1TAS1R3TAS1R1HPGDLMNA
SCHEMBL20658192 0.82 TAS1R3 (0.52) ALDH1A1TAS1R3TAS1R1HPGDLMNA
SCHEMBL1557472 0.81 SMN1; SMN2 (0.69) ALDH1A1TAS1R3TAS1R1NFE2L2HPGD
SCHEMBL1558819 0.81 SMN1; SMN2 (0.69) ALDH1A1TAS1R3TAS1R1NFE2L2HPGD
SCHEMBL1558821 0.81 SMN1; SMN2 (0.69) ALDH1A1TAS1R3TAS1R1NFE2L2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250143359-A1 COMPOUNDS THAT MODULATE GPR92 RECEPTOR ACTIVITY AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2025-05-08 US disclosed
US-20250127196-A1 COMPOUNDS THAT MODULATE FATTY ACID RECEPTOR ACTIVITY AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2025-04-24 US disclosed
EP-3229611-B1 COMPOUNDS THAT MODULATE FATTY ACID RECEPTOR ACTIVITY AND PET FOOD PRODUCTS CONTAINING THE SAME MARS INC (US) 2025-03-26 EP disclosed
US-12207673-B2 Compounds that modulate fatty acid receptor activity and pet food products containing the same MARS, INCORPORATED (US) 2025-01-28 US disclosed
US-12207672-B2 Compounds that modulate GPR92 receptor activity and pet food products containing the same MARS, INCORPORATED (US) 2025-01-28 US disclosed
EP-4403042-A2 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME Mars, Incorporated (US) 2024-07-24 EP disclosed
EP-3229612-B1 USE OF FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS INC (US) 2024-06-26 EP disclosed
US-11185100-B2 Methods for modulating taste receptors MARS, INCORPORATED (US) 2021-11-30 US disclosed
US-11185100-B2 Methods for modulating taste receptors MARS, INCORPORATED (US) 2021-11-30 US disclosed
US-20210315244-A1 COMPOUNDS THAT MODULATE GPR92 RECEPTOR ACTIVITY AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2021-10-14 US disclosed
EP-3229612-A2 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME Mars, Incorporated (US) 2017-10-18 EP disclosed
EP-3229606-A2 METHODS FOR MODULATING TASTE RECEPTORS Mars, Incorporated (US) 2017-10-18 EP disclosed
EP-3229611-A2 COMPOUNDS THAT MODULATE FATTY ACID RECEPTOR ACTIVITY AND PET FOOD PRODUCTS CONTAINING THE SAME Mars, Incorporated (US) 2017-10-18 EP disclosed
WO-2016094702-A2 METHODS FOR MODULATING TASTE RECEPTORS MARS, INCORPORATED (US) 2016-06-16 WO disclosed
WO-2016094682-A2 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2016-06-16 WO disclosed
WO-2016094682-A2 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2016-06-16 WO disclosed
WO-2016094726-A2 COMPOUNDS THAT MODULATE FATTY ACID RECEPTOR ACTIVITY AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2016-06-16 WO disclosed
WO-2016094690-A1 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2016-06-16 WO disclosed
WO-2016094690-A1 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2016-06-16 WO disclosed
WO-2016094702-A2 METHODS FOR MODULATING TASTE RECEPTORS MARS, INCORPORATED (US) 2016-06-16 WO disclosed