SCHEMBL178250

SCHEMBL178250

O=C(Nc1ccc(-c2cnc(CCNS(=O)(=O)CF)s2)cc1)Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.43
P2RY1 P47900 1/20 0.42
DGAT1 O75907 2/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
MAPT P10636 1/20 0.41
NTRK1 P04629 3/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
KDR P35968 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
NAMPT P43490 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
BAZ1A Q9NRL2 1/20 0.38
MTOR P42345 1/20 0.38
CA4 P22748 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL178117 0.90 EPHX2 (0.45) EPHX2P2RY1DGAT1CA12CA1
SCHEMBL15022122 0.89 EPHX2 (0.44) EPHX2P2RY1DGAT1CA12CA1
SCHEMBL174942 0.89 DGAT1 (0.48) EPHX2DGAT1KDRNAMPT
SCHEMBL176236 0.84 DGAT1 (0.54) DGAT1CA12CA1CA2CA9
SCHEMBL15021989 0.82 EPHX2 (0.47) EPHX2P2RY1DGAT1CA12CA1
SCHEMBL162613 0.82 TRPV1 (0.47) DGAT1HDAC1HDAC6TRPV1MEN1
SCHEMBL178251 0.80 NTRK1 (0.45) EPHX2P2RY1DGAT1CA12CA1
SCHEMBL15021905 0.80 DGAT1 (0.48) DGAT1KDRNAMPT
SCHEMBL175408 0.79 DGAT1 (0.48) DGAT1KDRNAMPT
SCHEMBL161990 0.78 DGAT1 (0.51) DGAT1MAPTNTRK1KDRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed