SCHEMBL17826910

SCHEMBL17826910

CN(C)c1ccc2[nH]cc(C(N)CNC(=O)OC(C)(C)C)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 0.42
MAPT P10636 9/20 0.42
MEN1 O00255 8/20 0.42
L3MBTL1 Q9Y468 8/20 0.42
ALDH1A1 P00352 6/20 0.42
TDP1 Q9NUW8 4/20 0.42
MAPK1 P28482 3/20 0.42
MCL1 Q07820 3/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
PTGS2 P35354 1/20 0.39
CTSL P07711 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
TRPV1 Q8NER1 2/20 0.36
CAPN1 P07384 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15944117 0.86 NR4A2 (0.43) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL3334684 0.85 AAK1 (0.45) MTNR1AMTNR1BCTSLCTSSCTSK
SCHEMBL3331422 0.84 MTNR1A (0.57) KMT2AMAPTMEN1ALDH1A1TDP1
SCHEMBL15944824 0.82 MTNR1A (0.39) KMT2AMAPTMEN1GAAMTNR1A
SCHEMBL13301913 0.82 MAPT (0.49) KMT2AMAPTMEN1L3MBTL1ALDH1A1
SCHEMBL13301912 0.79 AAK1 (0.45) MTNR1AMTNR1B
SCHEMBL13302029 0.75 HDAC10 (0.35) MAPK1MTNR1AMTNR1B
SCHEMBL17826908 0.73 MTNR1A (0.54) MTNR1AMTNR1BTRPV1
Trimethylammonium SCHEMBL9095683 0.72 MAPT (0.47) KMT2AMAPTMEN1L3MBTL1ALDH1A1
SCHEMBL3333209 0.72 NR4A2 (0.44) MTNR1AMTNR1BTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121601-B1 NOVEL INDOLE DERIVATIVES, METHODS FOR PREPARING SAME, AND USE THEREOF PARTICULARLY AS ANTIBACTERIAL AGENTS Université Joseph Fourier (FR) 2016-06-15 EP disclosed