SCHEMBL17835012

SCHEMBL17835012

Brc1ccc2c(c1)C1(c3cc(Br)ccc3-2)c2ccccc2N(c2cc(-c3cccnc3)cc(-c3cccnc3)c2)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.41
CYP11B2 P19099 4/20 0.41
PDK2 Q15119 2/20 0.40
USP8 P40818 1/20 0.37
MAPT P10636 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2A6 P11509 1/20 0.34
TDP2 O95551 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
GLO1 Q04760 1/20 0.33
CYP19A1 P11511 4/20 0.33
CYP17A1 P05093 1/20 0.33
HSP90AA1 P07900 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA3 P34903 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19754289 0.87 PDK2 (0.38) PDK2ALDH1A1EGLN1
SCHEMBL15084749 0.84 CYP11B1 (0.41) CYP11B1CYP11B2PDK2USP8MAPT
SCHEMBL17835006 0.84 CYP11B2 (0.44) CYP11B1CYP11B2PDK2CYP19A1CYP17A1
SCHEMBL12126537 0.77 PDK2 (0.42) PDK2ALDH1A1CYP1A2CYP3A4TDP2
SCHEMBL17835066 0.76 PDK2 (0.40) PDK2NPC1RAB9AALDH1A1TDP2
SCHEMBL20689955 0.75 ALDH1A1 (0.38) NPC1RAB9AALDH1A1CYP1A2CYP3A4
SCHEMBL19007133 0.75 PDK2 (0.43) PDK2MAPTALDH1A1CYP1A2CYP3A4
SCHEMBL29461269 0.75 PDK2 (0.43) PDK2MAPTALDH1A1CYP1A2CYP3A4
SCHEMBL20689959 0.75 HTT (0.38) MAPTALDH1A1CYP1A2CYP3A4CYP2A6
SCHEMBL13085651 0.74 EGLN1 (0.38) PDK2NPC1RAB9AALDH1A1TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10683453-B2 Organic compounds with soluble groups MERCK PATENT GMBH (DE) 2020-06-16 US disclosed
EP-3230403-B1 ORGANIC COMPOUNDS WITH SOLUBLE GROUPS MERCK PATENT GMBH (DE) 2019-10-09 EP disclosed
US-20170369773-A1 ORGANIC COMPOUNDS WITH SOLUBLE GROUPS UDC IRELAND LIMITED (IE) 2017-12-28 US disclosed
WO-2016091353-A1 ORGANIC COMPOUNDS WITH SOLUBLE GROUPS MERCK PATENT GMBH (DE) 2016-06-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170369773-A1 ORGANIC COMPOUNDS WITH SOLUBLE GROUPS SLCO4C1, SLCO1B3, SLCO2B1 CYP11B1 348/4885CYP11B2 228/4885PDK2 2619/4885
US-10683453-B2 Organic compounds with soluble groups SLCO4C1, SLCO1B3, SLCO2B1 CYP11B1 348/4885CYP11B2 228/4885PDK2 2619/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.