SCHEMBL17837308

SCHEMBL17837308

C=CCOC(=O)C1(C(N)C(=O)Oc2ccc(F)cc2)CCCCC1=O

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 6/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP3A4 P08684 3/20 0.32
TSHR P16473 3/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP2C9 P11712 2/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
FAAH O00519 1/20 0.30
GRM2 Q14416 1/20 0.30
GRM3 Q14832 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17837301 0.90 CA1 (0.39) CYP2C19KMT2AMEN1CYP2D6CYP3A4
SCHEMBL17837267 0.90 CYP3A4 (0.39) CYP2C19KMT2AMEN1CYP2D6CYP3A4
SCHEMBL17837292 0.78 CYP3A4 (0.39) CYP2C19CYP3A4TSHRALDH1A1CYP2C9
SCHEMBL17837304 0.77 CYP2C19 (0.32) CYP2C19CYP3A4TSHRALDH1A1CYP2C9
SCHEMBL17837309 0.76 FAAH (0.36) KMT2ATSHRALDH1A1POLBMAPK1
SCHEMBL17837312 0.74 CYP2C19 (0.35) CYP2C19KMT2AMEN1CYP2D6CYP3A4
SCHEMBL17854733 0.67 FAAH (0.38) CYP2C19KMT2ATSHRPOLBFAAH
SCHEMBL17837303 0.65 FAAH (0.38) KMT2AMEN1TSHRALDH1A1CYP2C9
SCHEMBL14498565 0.65 ALDH1A1 (0.33) CYP3A4TSHRALDH1A1POLB
SCHEMBL17837269 0.65 FAAH (0.38) CYP3A4ALDH1A1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11377396-B2 Enantioselective synthesis of α-quaternary Mannich adducts by palladium-catalyzed allylic alkylation CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-07-05 US disclosed
US-20200157020-A1 ENANTIOSELECTIVE SYNTHESIS OF ALPHA-QUATERNARY MANNICH ADDUCTS BY PALLADIUM-CATALYZED ALLYLIC ALKYLATION CALIFORNIA INSTITUTE OF TECHNOLOGY 2020-05-21 US disclosed
US-10421696-B2 Enantioselective synthesis of α-quaternary mannich adducts by palladium-catalyzed allylic alkylation CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2019-09-24 US disclosed
US-20160176773-A1 ENANTIOSELECTIVE SYNTHESIS OF alpha-QUATERNARY MANNICH ADDUCTS BY PALLADIUM-CATALYZED ALLYLIC ALKYLATION CALIFORNIA INSTITUTE OF TECHNOLOGY 2016-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11377396-B2 Enantioselective synthesis of α-quaternary Mannich adducts by palladium-catalyzed allylic alkylation ALG8, MANBA, MAN2A1 CYP2C19 492/4885KMT2A 214/4885MEN1 117/4885
US-10421696-B2 Enantioselective synthesis of α-quaternary mannich adducts by palladium-catalyzed allylic alkylation ALG8, MANBA, MAN2A1 CYP2C19 492/4885KMT2A 214/4885MEN1 117/4885
US-20160176773-A1 ENANTIOSELECTIVE SYNTHESIS OF alpha-QUATERNARY MANNICH ADDUCTS BY PALLADIUM-CATALYZED ALLYLIC ALKYLATION ALG8, MANBA, MAN2A1 CYP2C19 651/4885KMT2A 245/4885MEN1 92/4885
US-20200157020-A1 ENANTIOSELECTIVE SYNTHESIS OF ALPHA-QUATERNARY MANNICH ADDUCTS BY PALLADIUM-CATALYZED ALLYLIC ALKYLATION ALG8, MANBA, MAN2A1 CYP2C19 651/4885KMT2A 245/4885MEN1 92/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.