SCHEMBL17844309

SCHEMBL17844309

COc1cc(C(=O)O)ccc1OCCc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.65
PDE4B Q07343 3/20 0.65
PDE4C Q08493 3/20 0.65
PDE4D Q08499 3/20 0.65
TSHR P16473 1/20 0.64
CA12 O43570 1/20 0.61
CA1 P00915 1/20 0.61
CA2 P00918 1/20 0.61
CA4 P22748 1/20 0.61
CA6 P23280 1/20 0.61
CA7 P43166 1/20 0.61
TPMT P51580 1/20 0.61
CA9 Q16790 1/20 0.61
CA14 Q9ULX7 1/20 0.61
TTR P02766 1/20 0.58
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
MRGPRX4 Q96LA9 2/20 0.58
HPGD P15428 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30622576 1.00 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL8890661 0.94 PDE4A (0.73) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL17844306 0.89 NPC1 (0.59) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL8122418 0.86 TSHR (0.78) TSHRCA12CA1CA2CA4
SCHEMBL8085474 0.86 TSHR (0.78) TSHRCA12CA1CA2CA4
SCHEMBL7153812 0.86 PDE4A (0.81) PDE4APDE4BPDE4CPDE4DCA12
SCHEMBL242563 0.85 MRGPRX4 (0.77) TSHRCA12CA1CA2CA4
SCHEMBL21614005 0.85 TSHR (0.76) TSHRCA12CA1CA2CA4
SCHEMBL5492174 0.85 TSHR (0.76) TSHRCA12CA1CA2CA4
SCHEMBL6583889 0.84 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233847-A1 AMIDO THIADIAZOLE DERIVATIVES AS NADPH OXIDASE INHIBITORS GenKyoTex Suisse SA (CH) 2017-10-25 EP disclosed
WO-2016098005-A1 AMIDO THIADIAZOLE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2016-06-23 WO disclosed