SCHEMBL17844741

SCHEMBL17844741

C=CCOC[C@@H](OC(=O)NC(C)(C)C)c1cccc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
SLC6A2 P23975 2/20 0.34
AOC3 Q16853 1/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
ITGA5 P08648 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
SLC6A4 P31645 1/20 0.34
CHRNA3 P32297 1/20 0.34
CYP2C19 P33261 1/20 0.34
HRH1 P35367 1/20 0.34
CHRNA7 P36544 1/20 0.34
OPRK1 P41145 1/20 0.34
CHRNA4 P43681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27741031 0.86 MAPT (0.39) MAPTMEN1KMT2ACYP2C19ALDH1A1
SCHEMBL27720282 0.86 MAPT (0.39) MAPTMEN1KMT2ACYP2C19ALDH1A1
SCHEMBL17844812 0.83 MAPT (0.37) MAPTMEN1KMT2ASLC6A2SLC6A4
SCHEMBL28076433 0.82 MAPT (0.46) MAPTMEN1KMT2AHPGDALOX15
SCHEMBL17844814 0.82 AOC3 (0.39) MEN1KMT2AAOC3IDO1CYP2D6
SCHEMBL17844781 0.82 AOC3 (0.39) MEN1KMT2AAOC3IDO1CYP2D6
SCHEMBL27726392 0.80 MAPT (0.44) MAPTHPGDALOX15SLC6A2AOC3
SCHEMBL27747207 0.80 MAPT (0.44) MAPTHPGDALOX15SLC6A2AOC3
SCHEMBL27955103 0.80 MAPT (0.44) MAPTHPGDALOX15SLC6A2AOC3
SCHEMBL28625095 0.75 MAPT (0.42) MAPTHPGDALOX15SLC6A2AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016095088-A1 ERK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed