SCHEMBL17844812

SCHEMBL17844812

C=CCOC[C@@H](OC(=O)NC(C)(C)C)c1ccc(Cl)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
SLC6A4 P31645 10/20 0.34
SLC6A2 P23975 9/20 0.34
SLC6A3 Q01959 9/20 0.34
CYP1A2 P05177 4/20 0.33
CYP3A4 P08684 4/20 0.33
CYP2D6 P10635 4/20 0.33
CYP2C9 P11712 4/20 0.33
CYP2C19 P33261 4/20 0.33
KCNH2 Q12809 2/20 0.33
FFAR1 O14842 2/20 0.33
ANO1 Q5XXA6 1/20 0.33
POLB P06746 1/20 0.33
APEX1 P27695 1/20 0.33
HTT P42858 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844741 0.83 MAPT (0.39) MAPTALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL27720282 0.80 MAPT (0.39) MAPTALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL27741031 0.80 MAPT (0.39) MAPTALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL17846143 0.73 MAPT (0.39) MAPTALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL17844773 0.73 MEN1 (0.40) MAPTALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL19348965 0.73 MEN1 (0.40) MAPTALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL17844757 0.72 HTR2C (0.34) MAPTALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL20204243 0.72 HTR2C (0.34) MAPTALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL28793493 0.70 MDM2 (0.37) MAPTALDH1A1SLC6A2SLC6A3POLB
SCHEMBL27952278 0.69 LMNA (0.40) ALDH1A1SLC6A3POLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016095088-A1 ERK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed