SCHEMBL17844922

SCHEMBL17844922

O=C(O)N1CCN(c2nc(F)cc3ccc(F)cc23)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
HSD17B10 Q99714 1/20 0.41
PDGFRB P09619 1/20 0.40
SMO Q99835 1/20 0.39
KRAS P01116 1/20 0.39
HTT P42858 3/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
MAPT P10636 2/20 0.38
GALR2 O43603 1/20 0.38
TP53 P04637 3/20 0.38
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844916 0.84 HCAR2 (0.46) KDM4EHSD17B10PDGFRBKRAS
SCHEMBL17861366 0.81 GRIA1 (0.49) KDM4EHTTLMNASMN1; SMN2MAPT
SCHEMBL17861456 0.77 HRH4 (0.49) ABL1
SCHEMBL28164415 0.76 HTT (0.44) KDM4EHSD17B10HTTSMN1; SMN2TSHR
Hydrochloric Acid SCHEMBL17845014 0.75 HRH4 (0.48) ABL1
SCHEMBL5826334 0.75 MTNR1B (0.49) KDM4EHSD17B10KMT2ASMN1; SMN2MAPT
SCHEMBL5506348 0.74 SMAD3 (0.56) KDM4EHSD17B10PDGFRBKMT2AMAPT
SCHEMBL17844946 0.72 MAPT (0.41) HTTLMNAMAPTTSHR
SCHEMBL17845020 0.72 MAPT (0.41) HTTKMT2ALMNAMAPTTSHR
SCHEMBL22442358 0.71 MGLL (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233827-A1 ANTIBACTERIAL COMPOUNDS HAVING BROAD SPECTRUM OF ACTIVITY Aziende Chimiche Riunite Angelini Francesco A.C.R. (IT) 2017-10-25 EP disclosed
WO-2016096686-A1 ANTIBACTERIAL COMPOUNDS HAVING BROAD SPECTRUM OF ACTIVITY AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A. (IT) 2016-06-23 WO disclosed