SCHEMBL17847356

SCHEMBL17847356

CC(=O)NS(=O)(=O)c1cccc(CN(CCc2ccc(Br)cc2)C2CCN(C3=CN(N)NN3)CC2)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHIT1 Q13231 13/20 0.38
CHIA Q9BZP6 13/20 0.38
KCNH2 Q12809 9/20 0.38
CHI3L1 P36222 1/20 0.36
MEN1 O00255 5/20 0.35
KMT2A Q03164 5/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17838860 0.81 CHIT1 (0.45) CHIT1CHIAKCNH2
SCHEMBL17847353 0.79 MEN1 (0.41) CHIT1CHIAKCNH2CHI3L1MEN1
SCHEMBL17847364 0.76 CHIT1 (0.50) CHIT1CHIAKCNH2CHI3L1
SCHEMBL17838827 0.73 KMT2A (0.47) CHIT1CHIAMEN1KMT2AALDH1A1
SCHEMBL17838868 0.72 CHIT1 (0.48) CHIT1CHIAKCNH2
SCHEMBL17847361 0.72 CHIT1 (0.49) CHIT1CHIAKCNH2
SCHEMBL17853346 0.72 PPARG (0.43) ALDH1A1
Hydrochloric Acid SCHEMBL17838856 0.71 PPARG (0.43) ALDH1A1
SCHEMBL17838879 0.69 STS (0.48) MEN1KMT2A
SCHEMBL17847358 0.68 CHIT1 (0.51) CHIT1CHIAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233832-A1 SUBSTITUTED AMINO TRIAZOLES USEFUL AS ACIDIC MAMMALIAN CHITINASE INHIBITORS ONCOARENDI THERAPEUTICS S.A. (PL) 2017-10-25 EP disclosed
WO-2016099311-A1 SUBSTITUTED AMINO TRIAZOLES USEFUL AS ACIDIC MAMMALIAN CHITINASE INHIBITORS OncoArendi Therapeutics Sp. z o.o. (PL) 2016-06-23 WO disclosed