SCHEMBL17847358

SCHEMBL17847358

NN1C=C(N2CCC(N(CCc3ccc(Cl)cc3)Cc3cccc(-c4nnn[nH]4)c3)CC2)NN1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHIT1 Q13231 20/20 0.51
CHIA Q9BZP6 20/20 0.51
KCNH2 Q12809 16/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17838891 0.83 CHIT1 (0.58) CHIT1CHIAKCNH2
SCHEMBL17838822 0.81 CHIT1 (0.49) CHIT1CHIAKCNH2
SCHEMBL17853471 0.76 CHIT1 (0.45) CHIT1CHIAKCNH2
SCHEMBL17847361 0.73 CHIT1 (0.49) CHIT1CHIAKCNH2
SCHEMBL17838873 0.71 CHIT1 (0.57) CHIT1CHIAKCNH2
SCHEMBL16825703 0.69 CHIT1 (0.74) CHIT1CHIAKCNH2
Hydrochloric Acid SCHEMBL18129160 0.69 CHIT1 (0.73) CHIT1CHIAKCNH2
SCHEMBL17847356 0.68 CHIT1 (0.38) CHIT1CHIAKCNH2
SCHEMBL21674338 0.68 CHIT1 (0.64) CHIT1CHIAKCNH2
SCHEMBL17838882 0.68 CHIT1 (0.58) CHIT1CHIAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233832-A1 SUBSTITUTED AMINO TRIAZOLES USEFUL AS ACIDIC MAMMALIAN CHITINASE INHIBITORS ONCOARENDI THERAPEUTICS S.A. (PL) 2017-10-25 EP disclosed
WO-2016099311-A1 SUBSTITUTED AMINO TRIAZOLES USEFUL AS ACIDIC MAMMALIAN CHITINASE INHIBITORS OncoArendi Therapeutics Sp. z o.o. (PL) 2016-06-23 WO disclosed