SCHEMBL17848558

SCHEMBL17848558

CC(=O)N(C)C1(C)CCN(C(=O)O)CC1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.37
OPRL1 P41146 2/20 0.37
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
CYP2C19 P33261 1/20 0.30
FFAR3 O14843 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17848671 0.75 USP2 (0.47) USP2ALDH1A1
SCHEMBL28379744 0.75 CTSD (0.34) USP2
SCHEMBL15759336 0.73 FFAR3 (0.38) OPRM1USP2ALDH1A1MAPK1CYP2C19
SCHEMBL20738595 0.73 OPRM1 (0.39) OPRM1OPRL1CYP2C19FFAR3
SCHEMBL20738603 0.73 OPRM1 (0.39) OPRM1OPRL1ALDH1A1CYP2C19FFAR3
SCHEMBL19641323 0.72 FFAR3 (0.39) USP2ALDH1A1MAPK1CYP2C19FFAR3
SCHEMBL4539328 0.72 OPRM1 (0.32) OPRM1OPRL1
SCHEMBL3646525 0.72 OPRM1 (0.32) OPRM1OPRL1
SCHEMBL24272639 0.72 OPRM1 (0.38) OPRM1OPRL1ALDH1A1FFAR3
SCHEMBL14501954 0.72 OPRM1 (0.38) OPRM1OPRL1ALDH1A1FFAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed