SCHEMBL17848973

SCHEMBL17848973

CC(C)Oc1nc2ccccc2nc1Cl

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.52
MAPT P10636 4/20 0.49
L3MBTL1 Q9Y468 4/20 0.49
ATM Q13315 3/20 0.49
TSHR P16473 2/20 0.42
KDM4E B2RXH2 5/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
PKM P14618 1/20 0.41
TLR8 Q9NR97 1/20 0.41
NPSR1 Q6W5P4 2/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
GAA P10253 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17848984 0.79 ALDH1A1 (0.51) TDP1MAPTL3MBTL1ATMKDM4E
SCHEMBL805035 0.78 L3MBTL1 (0.51) MAPTL3MBTL1ATMTSHRKDM4E
SCHEMBL2178510 0.78 TDP1 (0.58) TDP1MAPTL3MBTL1TSHRKDM4E
SCHEMBL789181 0.77 KDM4E (0.51) MAPTL3MBTL1ATMTSHRKDM4E
SCHEMBL30829251 0.77 TDP1 (0.47) TDP1MAPTL3MBTL1ATMKDM4E
SCHEMBL13956255 0.74 L3MBTL1 (0.50) TDP1MAPTL3MBTL1ATMTSHR
SCHEMBL17184396 0.73 NPC1 (0.50) MAPTL3MBTL1KDM4EMEN1KMT2A
SCHEMBL2422773 0.73 HDAC1 (0.38) TDP1KDM4EHRH4GAA
SCHEMBL13966259 0.73 ATM (0.56) TDP1MAPTL3MBTL1ATMTSHR
SCHEMBL12410057 0.73 TDP1 (0.52) TDP1MAPTL3MBTL1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100101-A1 RUTHENIUM-BASED METATHESIS PRE-CATALYST COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed
WO-2016100101-A1 RUTHENIUM-BASED METATHESIS PRE-CATALYST COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed