SCHEMBL17849191

SCHEMBL17849191

CC(C)(C#N)c1ccc(C(=N)c2c(Nc3c(F)cccc3F)c(Cl)c[nH]c2=O)cc1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.34
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623476 0.86
SCHEMBL16623450 0.82 NPC1 (0.32) MAPT
SCHEMBL16623588 0.80 SYK (0.34)
SCHEMBL16726696 0.78 HDAC6 (0.41) RAB9A
SCHEMBL17849220 0.77 MT-CO2 (0.35)
SCHEMBL16726665 0.77 ALDH2 (0.33)
SCHEMBL16623587 0.76 ROCK1 (0.39) BRAFMAPTRAB9ANPSR1
SCHEMBL17849213 0.75 POLB (0.35) MAPT
SCHEMBL17849208 0.75 HDAC6 (0.33) MAPT
SCHEMBL16623547 0.75 SYK (0.36) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed