SCHEMBL17849220

SCHEMBL17849220

N=C(c1ccc(NCCO)cc1)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 1/20 0.35
HDAC6 Q9UBN7 1/20 0.34
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16726696 0.88 HDAC6 (0.41) HDAC6KDM4E
SCHEMBL17849206 0.82 ALDH1A1 (0.40) KDM4E
SCHEMBL16726665 0.82 ALDH2 (0.33)
SCHEMBL16623450 0.81 NPC1 (0.32)
SCHEMBL17849208 0.79 HDAC6 (0.33) HDAC6
SCHEMBL16623547 0.79 SYK (0.36) KDM4E
SCHEMBL16623588 0.79 SYK (0.34)
SCHEMBL16726674 0.79 PRKAB2 (0.35)
SCHEMBL17849211 0.78 L3MBTL1 (0.38) HDAC6KDM4E
SCHEMBL16623587 0.78 ROCK1 (0.39) HDAC6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed