SCHEMBL17849239

SCHEMBL17849239

CC(=O)Nc1ccc(C(=N)c2c(Nc3c(F)cccc3F)cc[nH]c2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.38
EGFR P00533 7/20 0.38
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC2 Q92769 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PARP1 P09874 1/20 0.35
IDO1 P14902 1/20 0.35
CACNA1B Q00975 1/20 0.35
APBA1 Q02410 1/20 0.35
TP53 P04637 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623511 0.84 TYK2 (0.38) PARP1JAK2
SCHEMBL16623558 0.83 PARP1 (0.34) PARP1
SCHEMBL16623596 0.82 HDAC6 (0.34) EGFRPARP1
SCHEMBL16623580 0.82 PARP1 (0.34) SMN1; SMN2EGFRRAB9AALDH1A1PARP1
SCHEMBL16726656 0.80 PTGS2 (0.33) PARP1
SCHEMBL17849218 0.79 HDAC6 (0.40) SMN1; SMN2ALDH1A1PARP1
SCHEMBL18052621 0.79 BRD4 (0.34) EGFRPARP1
SCHEMBL16623485 0.78 PARP1 (0.37) NPC1RAB9APARP1KMT2A
SCHEMBL16623583 0.78 EGFR (0.42) HDAC1EGFRHDAC3HDAC2ALDH1A1
SCHEMBL16726648 0.78 KDR (0.33) PARP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed