SCHEMBL16623596

SCHEMBL16623596

N=C(c1ccc(NCCNO)cc1)c1c(Nc2c(F)cccc2F)cc[nH]c1=O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.34
EGFR P00533 2/20 0.32
PRSS1 P07477 7/20 0.31
PARP1 P09874 1/20 0.31
F2 P00734 2/20 0.30
PRSS2 P07478 2/20 0.30
PRSS3 P35030 2/20 0.30
TMPRSS6 Q8IU80 2/20 0.30
ST14 Q9Y5Y6 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623558 0.82 PARP1 (0.34) PARP1
SCHEMBL17849239 0.82 HDAC1 (0.46) EGFRPARP1
SCHEMBL16623511 0.81 TYK2 (0.38) PARP1
SCHEMBL17849218 0.80 HDAC6 (0.40) HDAC6PARP1
SCHEMBL16726648 0.79 KDR (0.33) PARP1
SCHEMBL16726656 0.79 PTGS2 (0.33) PRSS1PARP1
SCHEMBL16623601 0.77 PRSS1 (0.37) EGFRPRSS1PRSS2PRSS3
SCHEMBL16623503 0.76 EGFR (0.35) EGFRPARP1
SCHEMBL17849238 0.76 L3MBTL1 (0.38) HDAC6EGFRPARP1
SCHEMBL18052621 0.76 BRD4 (0.34) EGFRPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed