SCHEMBL17850404

SCHEMBL17850404

COc1cc(-n2cc(-c3n[nH]c4ccccc34)[nH]2)ccc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 6/20 0.45
NPC1 O15118 1/20 0.42
CASP3 P42574 1/20 0.42
RAB9A P51151 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAP2K4 P45985 2/20 0.42
MAPK1 P28482 1/20 0.42
MAPKAPK3 Q16644 1/20 0.42
MAPK6 Q16659 1/20 0.42
CTNNB1 P35222 1/20 0.40
WNT3A P56704 1/20 0.40
CHEK1 O14757 2/20 0.39
FGFR1 P11362 2/20 0.39
CDK4 P11802 2/20 0.39
CCNA2 P20248 2/20 0.39
CCND1 P24385 2/20 0.39
CDK2 P24941 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9951964 0.82 STIM1 (0.41) ITKNPC1CASP3RAB9ASENP8
SCHEMBL9952459 0.73 NOTUM (0.45) ITKNPC1CASP3RAB9ASENP8
SCHEMBL9953228 0.71 NPC1 (0.39) ITKNPC1CASP3RAB9ASENP8
SCHEMBL9952540 0.70 KDM4E (0.45) NPC1CASP3RAB9ASENP8SENP7
SCHEMBL1597216 0.70 CHEK1 (0.51) ITKNPC1CASP3RAB9ASENP8
SCHEMBL1597212 0.70 CHEK1 (0.51) ITKNPC1CASP3RAB9ASENP8
SCHEMBL10208055 0.65 ALDH1A1 (0.49) ALDH1A1HPGDKDM4E
SCHEMBL31357524 0.65 MAP2K4 (0.60) ITKNPC1RAB9AMAP2K4MAPK1
SCHEMBL5822772 0.65 MAP2K4 (0.60) ITKNPC1RAB9AMAP2K4MAPK1
SCHEMBL2858040 0.64 CDK4 (0.60) NPC1RAB9AMAP2K4MAPK1MAPKAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed