SCHEMBL17855855

SCHEMBL17855855

FC1=CC=C(c2ccc(Cc3ccc(-c4ccc(F)cc4)c(F)c3)cc2F)CC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHKA P35790 1/20 0.35
GRM2 Q14416 4/20 0.35
HTR2A P28223 1/20 0.35
APP P05067 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
RARB P10826 1/20 0.32
MAOB P27338 2/20 0.32
DPP4 P27487 1/20 0.32
ABCB1 P08183 1/20 0.32
FDFT1 P37268 1/20 0.32
CNR1 P21554 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
MAOA P21397 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13624599 0.82 MAOB (0.44) CHKAGRM2HTR2AAPPCYP3A4
SCHEMBL19651371 0.69 FDFT1 (0.47) CHKAGRM2HTR2AAPPCYP3A4
SCHEMBL17900079 0.69 MAOB (0.41) CHKAGRM2HTR2AAPPCYP3A4
SCHEMBL16848650 0.67 RARB (0.51) CHKAGRM2HTR2AAPPCYP3A4
SCHEMBL16848654 0.67 RARB (0.51) CHKAGRM2HTR2AAPPCYP3A4
SCHEMBL16748099 0.66 CYP17A1 (0.57) CHKAGRM2CYP3A4PDE3BPDE3A
SCHEMBL16922714 0.66 APP (0.53) GRM2APPMAOB
SCHEMBL15587742 0.66 AMY1A (0.39) GRM2PDE3BPDE3A
SCHEMBL19993271 0.65 PTGS1 (0.38) GRM2APPCYP3A4MAOBPTGS1
SCHEMBL16941050 0.65 PTGS1 (0.46) GRM2PDE3BPDE3ARARBMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016096081-A1 BIMESOGENIC COMPOUNDS AND MESOGENIC MEDIA MERCK PATENT GMBH (DE) 2016-06-23 WO disclosed