SCHEMBL17866258

SCHEMBL17866258

O=C(Nc1cnc(OCC(F)(F)F)c(-c2ccc(Cl)cc2)c1)Oc1ccno1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.47
KCNH2 Q12809 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
PTGS2 P35354 2/20 0.39
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CNR2 P34972 1/20 0.37
ROCK2 O75116 2/20 0.34
GAA P10253 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
CHEK1 O14757 1/20 0.33
IKBKB O14920 1/20 0.33
DCLK1 O15075 1/20 0.33
RPS6KA5 O75582 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2112861 0.85 CNR1 (0.52) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866251 0.84 CNR1 (0.47) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866268 0.83 CNR1 (0.47) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866261 0.83 CNR1 (0.47) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866284 0.83 CNR1 (0.48) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866289 0.83 MAPT (0.45) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866266 0.83 MAPT (0.45) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866263 0.82 CNR1 (0.46) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866280 0.82 CNR1 (0.46) CNR1KCNH2SCN5ASCN2ASCN10A
SCHEMBL17866260 0.82 CNR1 (0.44) CNR1KCNH2SCN5ASCN2ASCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627637-B1 N-PYRIDIN-3-YL OR N-PYRAZIN-2-YL CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2016-06-29 EP claimed