SCHEMBL17866262

SCHEMBL17866262

O=C(Nc1cnc(OCC(F)(F)F)c(-c2ccc(Cl)cc2)c1)Oc1ccc(O)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.47
MAPT P10636 5/20 0.42
NPSR1 Q6W5P4 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PTGS2 P35354 2/20 0.39
KCNH2 Q12809 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
EPHX2 P34913 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
DEGS1 O15121 1/20 0.36
CHEK1 O14757 1/20 0.35
IKBKB O14920 1/20 0.35
DCLK1 O15075 1/20 0.35
ROCK2 O75116 1/20 0.35
RPS6KA5 O75582 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17866268 0.87 CNR1 (0.47) CNR1MAPTNPSR1SMN1; SMN2PTGS2
SCHEMBL2117015 0.86 CNR1 (0.52) CNR1PTGS2KCNH2SCN5ASCN2A
SCHEMBL17866263 0.86 CNR1 (0.46) CNR1MAPTNPSR1SMN1; SMN2PTGS2
SCHEMBL17866251 0.86 CNR1 (0.47) CNR1MAPTNPSR1SMN1; SMN2PTGS2
SCHEMBL17866283 0.85 CNR1 (0.47) CNR1MAPTNPSR1SMN1; SMN2PTGS2
SCHEMBL17866270 0.83 CNR1 (0.45) CNR1MAPTNPSR1SMN1; SMN2PTGS2
SCHEMBL17866284 0.83 CNR1 (0.48) CNR1MAPTNPSR1SMN1; SMN2PTGS2
SCHEMBL17866266 0.83 MAPT (0.45) CNR1MAPTNPSR1SMN1; SMN2PTGS2
SCHEMBL17866254 0.83 MAPT (0.49) CNR1MAPTNPSR1SMN1; SMN2PTGS2
SCHEMBL17866258 0.81 CNR1 (0.47) CNR1MAPTNPSR1SMN1; SMN2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627637-B1 N-PYRIDIN-3-YL OR N-PYRAZIN-2-YL CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2016-06-29 EP claimed