SCHEMBL17870754

SCHEMBL17870754

CS(=O)(=O)CCn1c(=O)[nH]cc(-c2cccc(F)c2Cl)c1=O

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 2/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33
GNRHR P30968 2/20 0.31
CYP3A4 P08684 1/20 0.31
CNR1 P21554 2/20 0.31
CNR2 P34972 2/20 0.31
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17870766 0.93 KDM4E (0.32) CCNE2CCNE1CDK2GNRHRCYP3A4
SCHEMBL30178654 0.93 KDM4E (0.32) CCNE2CCNE1CDK2GNRHRCYP3A4
SCHEMBL30178288 0.88 CNR1 (0.35) CCNE2CCNE1CDK2CNR1CNR2
SCHEMBL30178581 0.82 CCNE2 (0.34) CCNE2CCNE1CDK2GNRHRJAK3
SCHEMBL21900258 0.80 APEX1 (0.42) CCNE2CCNE1CDK2GNRHRCYP3A4
SCHEMBL28645646 0.79 CHEK1 (0.38) GNRHRCYP3A4
SCHEMBL19873696 0.78 KDM4E (0.44) CCNE2CCNE1CDK2GNRHRCYP3A4
SCHEMBL30178432 0.77 CCNE2 (0.32) CCNE2CCNE1CDK2
SCHEMBL21900230 0.77 FPR1 (0.41) CCNE2CCNE1CDK2
SCHEMBL28641642 0.76 KDM4E (0.45) JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3237403-A1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS Galderma Research & Development (FR) 2017-11-01 EP disclosed
WO-2016102882-A1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS GALDERMA RESEARCH & DEVELOPMENT (FR) 2016-06-30 WO disclosed