SCHEMBL28645646

SCHEMBL28645646

COC(=O)CCn1c(=O)[nH]cc(-c2cccc(F)c2Cl)c1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.38
WEE1 P30291 1/20 0.38
KAT2B Q92831 2/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
CYP3A4 P08684 1/20 0.35
GNRHR P30968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28641642 0.89 KDM4E (0.45) KDM4EALDH1A1SMN1; SMN2
SCHEMBL21900258 0.86 APEX1 (0.42) CHEK1WEE1KDM4EALDH1A1CYP3A4
SCHEMBL19873696 0.82 KDM4E (0.44) CHEK1WEE1KAT2BKDM4EALDH1A1
SCHEMBL17870801 0.80 IDO1 (0.33) SMN1; SMN2
SCHEMBL19873965 0.80 JAK3 (0.37) KDM4EALDH1A1SMN1; SMN2GNRHR
SCHEMBL17870711 0.80 IDO1 (0.43)
SCHEMBL30178581 0.80 CCNE2 (0.34) KDM4EALDH1A1SMN1; SMN2GNRHR
SCHEMBL21900230 0.79 FPR1 (0.41) KDM4E
SCHEMBL17870754 0.79 CCNE2 (0.33) CYP3A4GNRHR
SCHEMBL19873988 0.77 APAF1 (0.36) CYP3A4GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3708566-B1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS GALDERMA RES & DEV (FR) 2023-02-08 EP disclosed
CN-107428744-B Novel heterocyclic compounds and their use in medicine and cosmetics 盖尔德马研究及发展公司 2021-09-24 CN disclosed