SCHEMBL17874036

SCHEMBL17874036

CCOC(=O)c1c(CBr)nc(-c2nccs2)nc1-c1ccccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.46
DBF4 Q9UBU7 2/20 0.46
GRM6 O15303 1/20 0.41
ALDH1A1 P00352 5/20 0.40
HPGD P15428 4/20 0.40
MAPT P10636 5/20 0.39
KDM4E B2RXH2 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 1/20 0.39
DHODH Q02127 2/20 0.38
KCNH2 Q12809 1/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 2/20 0.37
PDE2A O00408 1/20 0.37
PDE10A Q9Y233 1/20 0.37
MAPK1 P28482 2/20 0.37
ATM Q13315 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17479130 0.88 CDC7 (0.49) CDC7DBF4GRM6ALDH1A1HPGD
SCHEMBL17064231 0.86 KMT2A (0.40) ALDH1A1HPGDMAPTKDM4ERAB9A
SCHEMBL15516071 0.78 HDAC3 (0.41) CDC7DBF4MAPTKCNH2
SCHEMBL16237173 0.73 CTSA (0.41) DHODH
SCHEMBL17064250 0.73 HCRTR1 (0.39) MAPTPOLBDHODHKMT2A
SCHEMBL16237487 0.73 HDAC3 (0.43) CDC7DBF4DHODH
SCHEMBL17874029 0.72 SCN9A (0.37) HPGDRAB9ANPC1
SCHEMBL7839276 0.72 ALDH1A1 (0.39) CDC7DBF4ALDH1A1HPGDMAPT
SCHEMBL19894057 0.71 TSHR (0.54) ALDH1A1MAPTKDM4EL3MBTL1RAB9A
SCHEMBL8946850 0.70 KDM4E (0.62) CDC7DBF4GRM6ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016102438-A1 PROCESS FOR THE PREPARATION OF 4-PHENYL-5-ALKOXYCARBONYL-2-THIAZOL-2-YL-1,4-DIHYDROPYRIMIDINE ANALOGUES F. HOFFMANN-LA ROCHE AG (CH) 2016-06-30 WO disclosed