SCHEMBL17874231

SCHEMBL17874231

CCc1c(C)nc(O)c(C(=O)O)c1O

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 12/20 0.41
RXRA P19793 3/20 0.37
NR4A2 P43354 3/20 0.37
PDE4B Q07343 1/20 0.37
PDE4D Q08499 1/20 0.37
LDHA P00338 2/20 0.35
LDHB P07195 2/20 0.35
ADORA3 P0DMS8 1/20 0.34
HSD17B10 Q99714 1/20 0.32
ALDH1A1 P00352 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL668597 0.75 HSD17B10 (0.41) LDHALDHBHSD17B10ALDH1A1
SCHEMBL2805456 0.74 ADORA3 (0.45) P2RX3RXRANR4A2PDE4BPDE4D
SCHEMBL9784563 0.72 HCAR2 (0.38) RXRANR4A2PDE4BPDE4DADORA3
SCHEMBL31436370 0.70 HCAR2 (0.41) RXRANR4A2PDE4BPDE4DADORA3
SCHEMBL14183027 0.70 ADORA3 (0.50) PDE4DADORA3HSD17B10ALDH1A1L3MBTL1
SCHEMBL15316167 0.70 PDE10A (0.44) P2RX3PDE4BPDE4DLDHALDHB
SCHEMBL28677095 0.68 FASN (0.39) LDHALDHBHSD17B10ALDH1A1
SCHEMBL4117808 0.68 FASN (0.47) LDHALDHBHSD17B10ALDH1A1
SCHEMBL31643874 0.68 FASN (0.39) LDHALDHBHSD17B10ALDH1A1
SCHEMBL4126384 0.68 CYP3A4 (0.56) LDHALDHBHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016102493-A1 IMIDAZOPYRIDINE EZH2 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-06-30 WO disclosed