SCHEMBL17878205

SCHEMBL17878205

N#CC1(c2ccccc2C=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 2/20 0.43
THRB P10828 1/20 0.43
BLM P54132 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 3/20 0.36
TRIM24 O15164 2/20 0.36
TRIM33 Q9UPN9 2/20 0.36
TSHR P16473 1/20 0.36
IL4I1 Q96RQ9 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
OPRM1 P35372 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
CYP2A6 P11509 2/20 0.32
GAA P10253 1/20 0.32
IMPDH2 P12268 1/20 0.32
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21443604 0.89 MEN1 (0.36) KMT2ALMNAMEN1THRBBLM
SCHEMBL31459294 0.81 ALDH1A1 (0.36) ALDH1A1OPRM1
SCHEMBL10526403 0.80 OPRM1 (0.39) KMT2AMEN1ALDH1A1SMN1; SMN2OPRM1
SCHEMBL9878437 0.76 ADORA2A (0.34) ALDH1A1
SCHEMBL16767385 0.76 SRC (0.37) KMT2AMEN1ALDH1A1TSHRHPGD
SCHEMBL16767321 0.76 ERN1 (0.43) TDP1ALDH1A1OPRM1ERN1
SCHEMBL2050361 0.72 CA12 (0.38) KMT2ALMNAMEN1BLMTDP1
SCHEMBL1769351 0.72 HDAC4 (0.41) LMNAALDH1A1SMN1; SMN2OPRM1NPC1
SCHEMBL30929543 0.72 HDAC4 (0.41) LMNAALDH1A1SMN1; SMN2OPRM1NPC1
SCHEMBL6898 0.71 HTR2A (0.35) KMT2AMEN1ALDH1A1SMN1; SMN2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016106106-A2 FUSED HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-30 WO disclosed