SCHEMBL17895178

SCHEMBL17895178

O=C(Nc1cc(C(F)(F)F)ccn1)c1ccccn1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 4/20 0.60
RIOK2 Q9BVS4 1/20 0.54
EPAS1 Q99814 1/20 0.54
GRM4 Q14833 3/20 0.53
BRAF P15056 1/20 0.51
CES1 P23141 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
KMT2A Q03164 1/20 0.50
SORT1 Q99523 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
CASP1 P29466 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HSD17B10 Q99714 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
GRM5 P41594 1/20 0.48
PYGL P06737 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1968503 0.84 ALOX15 (0.60) RIOK2SORT1ALOX15TSHRCASP1
SCHEMBL30643207 0.82 EPAS1 (0.59) RIOK2EPAS1GRM4MEN1ALDH1A1
SCHEMBL16762179 0.81 EPAS1 (0.55) TLR7RIOK2EPAS1BRAFALDH1A1
SCHEMBL30362400 0.81 TRPV1 (0.57) RIOK2EPAS1MEN1ALDH1A1KMT2A
SCHEMBL28290705 0.80 KMT2A (0.71) TLR7GRM4BRAFCES1MEN1
SCHEMBL30360592 0.80 KMT2A (0.71) TLR7GRM4BRAFCES1MEN1
Formic Acid SCHEMBL30595912 0.80 ALOX15 (0.55) RIOK2EPAS1SORT1ALOX15TSHR
SCHEMBL15877592 0.80 GRM5 (0.48) RIOK2EPAS1MEN1ALDH1A1KMT2A
SCHEMBL13173412 0.79 TLR7 (0.54) TLR7GRM4BRAFCES1
SCHEMBL11483728 0.79 GRM4 (0.63) TLR7RIOK2GRM4TSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016106625-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-07-07 WO disclosed