SCHEMBL17899015

SCHEMBL17899015

COc1ccnc(C(=O)N[C@H]2CCCC[C@H](OC)[C@@H](OCC(C)C)[C@H](C)OC2=O)c1O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 4/20 0.33
TAS1R1 Q7RTX1 4/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PDE10A Q9Y233 1/20 0.31
ADORA2A P29274 1/20 0.31
TAS1R2 Q8TE23 2/20 0.30
HPGDS O60760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17899012 0.96 TAS1R3 (0.33) TAS1R3TAS1R1NPC1RAB9APDE10A
SCHEMBL15854921 0.94 TAS1R3 (0.33) TAS1R3TAS1R1NPC1RAB9APDE10A
SCHEMBL15861108 0.92 TAS1R3 (0.31) TAS1R3TAS1R1NPC1RAB9A
SCHEMBL15860583 0.92 TAS1R3 (0.33) TAS1R3TAS1R1NPC1RAB9AADORA2A
SCHEMBL19099682 0.92 TAS1R3 (0.34) TAS1R3TAS1R1NPC1RAB9APDE10A
SCHEMBL15861117 0.92 TAS1R3 (0.31) TAS1R3TAS1R1
SCHEMBL15861118 0.91 TAS1R3 (0.30) TAS1R3TAS1R1
SCHEMBL17899018 0.91 TAS1R3 (0.33) TAS1R3TAS1R1ADORA2A
SCHEMBL15844003 0.90 TAS1R3 (0.31) TAS1R3TAS1R1
SCHEMBL15854955 0.90 HPGDS (0.33) TAS1R3TAS1R1NPC1RAB9AHPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016109290-A1 MACROCYCLIC PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed
WO-2016109291-A1 USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed