SCHEMBL17907484

SCHEMBL17907484

COCOc1cccc(OCc2ccc(F)cc2)c1C=CC(=O)c1nc[nH]n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 2/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
AKR1C3 P42330 2/20 0.36
POLB P06746 1/20 0.36
PKM P14618 1/20 0.36
BLM P54132 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LTB4R Q15722 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
PLA2G1B P04054 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL754365 0.83 PPARG (0.49) BACE1MAOAMAOBKMT2AMEN1
SCHEMBL17907485 0.82 MAOB (0.37) MAOBKMT2AMEN1POLBPKM
SCHEMBL754366 0.73 MAPT (0.46) BACE1MAOAMAOBKMT2AMEN1
SCHEMBL754648 0.71 MAOB (0.46) BACE1MAOAMAOB
SCHEMBL10870465 0.64 PTGER1 (0.54) KMT2AMEN1PKMTDP1ALDH1A1
SCHEMBL10870470 0.64 PTGER1 (0.54) KMT2AMEN1PKMTDP1ALDH1A1
SCHEMBL27252704 0.64 MAPT (0.55) MAOAMAOBTDP1RAB9ANPC1
SCHEMBL14129787 0.64 MAOB (0.41) MAOAMAOBKMT2AMEN1ALDH1A1
SCHEMBL6035778 0.64 PTGER4 (0.60) ABCG2AKR1C3PKMALDH1A1
SCHEMBL6035782 0.64 PTGER4 (0.60) ABCG2AKR1C3PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3042894-A1 ANTIVIRAL AGENT SHIONOGI & CO., LTD. (JP) 2016-07-13 EP disclosed