SCHEMBL17907945

SCHEMBL17907945

CC(C)(C)OC(=O)Cn1c(C=CC(=O)O)cc2ccc(F)cc21

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
PLA2G7 Q13093 1/20 0.37
CCR2 P41597 1/20 0.35
NTRK1 P04629 1/20 0.35
CACNA1B Q00975 1/20 0.34
HK1 P19367 2/20 0.33
HKDC1 Q2TB90 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDO2 P48775 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
BRD4 O60885 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CDK9 P50750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907944 1.00 ALDH1A1 (0.37) ALDH1A1KDM4EPLA2G7CCR2NTRK1
SCHEMBL17907997 0.91 CACNA1B (0.40) ALDH1A1KDM4EPLA2G7CCR2NTRK1
SCHEMBL17907996 0.91 CACNA1B (0.40) ALDH1A1KDM4EPLA2G7CCR2NTRK1
SCHEMBL17907939 0.88 CCR9 (0.42) ALDH1A1KDM4ECCR2CACNA1BSMN1; SMN2
SCHEMBL17907937 0.88 CCR9 (0.42) ALDH1A1KDM4ECCR2CACNA1BSMN1; SMN2
SCHEMBL17907946 0.87 PDE5A (0.40) ALDH1A1KDM4ECCR2CACNA1BLMNA
SCHEMBL17907948 0.87 PDE5A (0.40) ALDH1A1KDM4ECCR2CACNA1BLMNA
SCHEMBL3553079 0.86 KDM4E (0.46) ALDH1A1KDM4ECCR2CACNA1BKMT2A
SCHEMBL3553083 0.86 KDM4E (0.46) ALDH1A1KDM4ECCR2CACNA1BKMT2A
SCHEMBL17907927 0.82 CACNA1B (0.44) ALDH1A1KDM4ECACNA1BMAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed