SCHEMBL17907997

SCHEMBL17907997

CC(C)(C)OC(=O)Cn1c(C=CC(=O)O)cc2cc(F)ccc21

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.40
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 2/20 0.38
HPGD P15428 1/20 0.38
PLA2G7 Q13093 1/20 0.37
CCR2 P41597 1/20 0.35
HK1 P19367 2/20 0.35
HKDC1 Q2TB90 2/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
F10 P00742 1/20 0.35
NTRK1 P04629 1/20 0.35
NR1I2 O75469 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
NR1H2 P55055 1/20 0.34
TDO2 P48775 1/20 0.33
ESR1 P03372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907996 1.00 CACNA1B (0.40) CACNA1BALDH1A1KDM4EHSD17B10HPGD
SCHEMBL17907944 0.91 ALDH1A1 (0.37) CACNA1BALDH1A1KDM4EHSD17B10PLA2G7
SCHEMBL17907945 0.91 ALDH1A1 (0.37) CACNA1BALDH1A1KDM4EHSD17B10PLA2G7
SCHEMBL17907928 0.89 CACNA1B (0.44) CACNA1BALDH1A1KDM4EHSD17B10MAPT
SCHEMBL17907927 0.89 CACNA1B (0.44) CACNA1BALDH1A1KDM4EHSD17B10MAPT
SCHEMBL17907951 0.88 TDP1 (0.41) CACNA1BALDH1A1KDM4EHPGDCCR2
SCHEMBL17907984 0.88 KDM4E (0.41) CACNA1BALDH1A1KDM4EHSD17B10HPGD
SCHEMBL17907953 0.88 TDP1 (0.41) CACNA1BALDH1A1KDM4EHPGDCCR2
SCHEMBL17907985 0.88 KDM4E (0.41) CACNA1BALDH1A1KDM4EHSD17B10HPGD
SCHEMBL3553079 0.86 KDM4E (0.46) CACNA1BALDH1A1KDM4ECCR2NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed