SCHEMBL17907951

SCHEMBL17907951

CC(C)(C)OC(=O)Cn1c(/C=C/C(=O)O)cc2cc(Cl)ccc21

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
CCR2 P41597 9/20 0.39
CACNA1B Q00975 1/20 0.39
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
THRB P10828 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TP53 P04637 1/20 0.33
ACLY P53396 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907953 1.00 TDP1 (0.41) TDP1CCR2CACNA1BKDM4EALDH1A1
SCHEMBL17907939 0.91 CCR9 (0.42) CCR2CACNA1BKDM4EALDH1A1HPGD
SCHEMBL17907937 0.91 CCR9 (0.42) CCR2CACNA1BKDM4EALDH1A1HPGD
SCHEMBL17907996 0.88 CACNA1B (0.40) CCR2CACNA1BKDM4EALDH1A1LMNA
SCHEMBL17907997 0.88 CACNA1B (0.40) CCR2CACNA1BKDM4EALDH1A1LMNA
SCHEMBL17907928 0.88 CACNA1B (0.44) TDP1CACNA1BKDM4EALDH1A1
SCHEMBL17907927 0.88 CACNA1B (0.44) TDP1CACNA1BKDM4EALDH1A1
SCHEMBL17907985 0.87 KDM4E (0.41) CCR2CACNA1BKDM4EALDH1A1THRB
SCHEMBL17907984 0.87 KDM4E (0.41) CCR2CACNA1BKDM4EALDH1A1THRB
SCHEMBL3553079 0.85 KDM4E (0.46) CCR2CACNA1BKDM4EALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed