SCHEMBL17907979

SCHEMBL17907979

O=C(O)NC1CCc2cc3ccc(Cl)cc3n2C1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
NOTUM Q6P988 1/20 0.34
CNR1 P21554 5/20 0.34
USP30 Q70CQ3 1/20 0.34
KRAS P01116 1/20 0.34
KMO O15229 2/20 0.33
CNR2 P34972 2/20 0.33
MAPK8 P45983 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRNA7 P36544 1/20 0.33
GRM5 P41594 1/20 0.33
F10 P00742 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907976 0.85 PTGDR2 (0.39) PTGDR2CHRNA7
SCHEMBL13279281 0.83 HTR2A (0.40) HTR2AHTR2CNOTUMCNR1CNR2
SCHEMBL14745400 0.72 USP30 (0.39) USP30KRASKMOKMT2A
SCHEMBL26912344 0.71 PTGDR2 (0.31) PTGDR2
SCHEMBL21028086 0.69 SMN1; SMN2 (0.39) HTR2AHTR2CKMT2A
SCHEMBL26913213 0.68 HTT (0.31) KRAS
SCHEMBL1534166 0.66 NOTUM (0.61) NOTUMCNR1USP30KMT2A
SCHEMBL17907974 0.66 NOS3 (0.41) PTGDR2HTR2AHTR2CCNR1CNR2
SCHEMBL17784836 0.66 NOTUM (0.64) PTGDR2HTR2ANOTUMCNR1KMT2A
SCHEMBL1800356 0.66 NOTUM (0.64) PTGDR2HTR2ANOTUMCNR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed